The library will operate on a duty schedule between 22 December 2025 and 4 January 2026. During this period, it will be possible to upload publications, but all other services will be suspended.
Kun, S.,
Begum, J.,
Kyriakis, E.,
Stamati, E. C. V.,
Barkas, T. A.,
Szennyes, E.,
Bokor, É.,
Szabó, E. K.,
Stravodimos, G. A.,
Sipos, Á.,
Docsa, T.,
Gergely, P.,
Moffatt, C.,
Patraskaki, M. S.,
Kokolaki, M. C.,
Gkerdi, A.,
Skamnaki, V. T.,
Leonidas, D. D.,
Somsák, L.,
Hayes, J. M.:
A multidisciplinary study of 3-(β-D-glucopyranosyl)-5-substituted-1,2,4-triazole derivatives as glycogen phosphorylase inhibitors: computation, synthesis, crystallography and kinetics reveal new potent inhibitors.
Eur. J. Med. Chem. 147, 266-278, 2018.
Gergely, P.,
Hodossy-Takács, E.,
Magyar, É.:
Beszámoló az MTA Debreceni Területi Bizottsága (a DAB) 2016. évi munkájáról.
Debr. szle. 25 (2), 244-259, 2017.
Bokor, É.,
Kyriakis, E.,
Solovou, T. G. A.,
Koppány, C.,
Kantsadi, A. L.,
Szabó, E. K.,
Szakács, A.,
Stravodimos, G. A.,
Docsa, T.,
Skamnaki, V. T.,
Zographos, S. E.,
Gergely, P.,
Leonidas, D. D.,
Somsák, L.:
Nanomolar Inhibitors of Glycogen Phosphorylase Based on β-d-Glucosaminyl Heterocycles: A Combined Synthetic, Enzyme Kinetic, and Protein Crystallography Study.
J. Med. Chem. 60 (22), 9251-9262, 2017.
Goyard, D.,
Kónya, B.,
Chajistamatiou, A. S.,
Chrysina, E. D.,
Leroy, J.,
Balzarin, S.,
Tournier, M.,
Tousch, D.,
Petit, P.,
Duret, C.,
Maurel, P.,
Somsák, L.,
Docsa, T.,
Gergely, P.,
Praly, J. P.,
Azay-Milhau, J.,
Vidal, S.:
Glucose-derived spiro-isoxazolines are anti-hyperglycemic agents against type 2 diabetes through glycogen phosphorylase inhibition.
Eur. J. Med. Chem. 108, 444-454, 2016.
Kantsadi, A. L.,
Bokor, É.,
Kun, S.,
Stravodimos, G. A.,
Chatzileontiadou, D. S. M.,
Leonidas, D. D.,
Juhász-Tóth, É.,
Szakács, A.,
Batta, G.,
Docsa, T.,
Gergely, P.,
Somsák, L.:
Synthetic, enzyme kinetic, and protein crystallographic studies of C-[béta]-D-glucopyranosyl pyrroles and imidazoles reveal and explain low nanomolar inhibition of human liver glycogen phosphorylase.
Eur. J. Med. Chem. 123, 737-745, 2016.
Goyard, D.,
Docsa, T.,
Gergely, P.,
Praly, J. P.,
Vidal, S.:
Synthesis of 4-amidomethyl-1-glucosyl-1,2,3-triazoles and evaluation as glycogen phosphorylase inhibitors.
Carbohydr. Res. 402, 245-251, 2015.
Czifrák, K.,
Páhi, A.,
Deák, S.,
Kiss-Szikszai, A.,
Kövér, K. E.,
Docsa, T.,
Gergely, P.,
Alexacou, K. M.,
Papakonstantinou, M.,
Leonidas, D. D.,
Zographos, S. E.,
Chrysina, E. D.,
Somsák, L.:
Glucopyranosylidene-spiro-iminothiazolidinone, a New Bicyclic Ring System: Synthesis, Derivatization, and Evaluation for Inhibition of Glycogen Phosphorylase by Enzyme Kinetic and Crystallographic Methods.
Bioorg. Med. Chem. 22 (15), 4028-4041, 2014.