The library will operate on a duty schedule between 22 December 2025 and 4 January 2026. During this period, it will be possible to upload publications, but all other services will be suspended.
Homolya, L.,
Mathomes, R. T.,
Varga, L.,
Docsa, T.,
Juhász, L.,
Hayes, J. M.,
Somsák, L.:
Synthesis, in silico and kinetics evaluation of N-(beta-D-glucopyranosyl)-2-arylimidazole-4(5)-carboxamides and N-(beta-D-glucopyranosyl)-4(5)-arylimidazole-2-carboxamides as glycogen phosphorylase inhibitors.
Int. J. Mol. Sci. 25 (9), 1-21, (article identifier: 4591), 2024.
József, J.,
Somsák, L.,
Tóth, M.,
Juhász, L.:
[2+2] Cycloadditions of Methylene exo-Glycals: Synthesis of Glycopyranosylidene-Spiro-Azetidine-2-ones (beta-Lactams) and Cyclobutanones.
Eur. J. Org. Chem. 26 (12), 1-10, (article identifier: 202201488), 2023.
Homolya, Á.,
Jedlóczki, I.,
Ábrahám, A.,
Somsák, L.,
Tóth, M.,
Juhász, L.:
Behaviour of some 1-C-acceptor-substituted glycals under azidohydroxylation conditions.
Carbohydr. Res. 529, 1-12, (article identifier: 108825), 2023.
Kun, S.,
Mathomes, R. T.,
Docsa, T.,
Somsák, L.,
Hayes, J. M.:
Design and Synthesis of 3-(β-D-Glucopyranosyl)-4-amino/4-guanidino Pyrazole Derivatives and Analysis of Their Glycogen Phosphorylase Inhibitory Potential.
Molecules. 28 (7), 1-19, (article identifier: 3005), 2023.
Bokor, É.,
Kecskés, D.,
Gombás, F.,
Fehér, A.,
Kardos, E.,
Dabian, A.,
Vonza, Z.,
Szennyes, E.,
Somsák, L.:
First representatives of C-glycosyl 1,2,4,5-tetrazines: synthesis of 3-beta-d-glucopyranosyl 1,2,4,5-tetrazines and their transformation into 3-beta-d-glucopyranosyl pyridazines.
New Journal of Chemistry 47 (1), 56-74, 2023.
Lázár, L.,
Tsagkarakou, A. S.,
Stravodimos, G. A.,
Kontopidis, G.,
Leffler, H.,
Nilsson, U. J.,
Somsák, L.,
Leonidas, D. D.:
Strong Binding of C-Glycosylic1,2-Thiodisaccharides to Galectin-3 - Enthalpy-Driven Affinity Enhancement by Water-Mediated Hydrogen Bonds.
Journal of Medicinal Chemistry 66 (17), 12420-12431, 2023.
Kiss, M.,
Timári, I.,
Barna, T.,
Mészáros, Z.,
Slámová, K.,
Bojarová, P.,
Křen, V.,
Hayes, J. M.,
Somsák, L.:
2-Acetamido-2-deoxy-d-glucono-1,5-lactone Sulfonylhydrazones: Synthesis and Evaluation as Inhibitors of Human OGA and HexB Enzymes.
Int. J. Mol. Sci. 23 (3), 1-18, (article identifier: 1037), 2022.
Kánya, N.,
Kun, S.,
Somsák, L.:
Glycopyranosylidene-Spiro-Morpholinones: Evaluation of the Synthetic Possibilities Based on Glyculosonamide Derivatives and a New Method for the Construction of the Morpholine Ring.
Molecules. 27 (22), 1-18, (article identifier: 7785), 2022.
Kacsir, I.,
Sipos, A.,
Bényei, A.,
Janka, E. A.,
Buglyó, P.,
Somsák, L.,
Bai, P.,
Bokor, É.:
Reactive Oxygen Species Production Is Responsible for Antineoplastic Activity of Osmium, Ruthenium, Iridium and Rhodium Half-Sandwich Type Complexes with Bidentate Glycosyl Heterocyclic Ligands in Various Cancer Cell Models.
Int. J. Mol. Sci. 23 (2), 1-39, (article identifier: 813), 2022.
Kaszás, T.,
Cservenyák, I.,
Juhász-Tóth, É.,
Kulcsár, A.,
Granatino, P.,
Nilsson, U. J.,
Somsák, L.,
Tóth, M.:
Coupling of N-tosylhydrazones with tetrazoles: synthesis of 2-beta-d-glycopyranosylmethyl-5-substituted-2H-tetrazole type glycomimetics.
Org. Biomol. Chem. 19 (3), 605-618, 2021.
Sipos, Á.,
Szennyes, E.,
Hajnal, É.,
Kun, S.,
Szabó, E. K.,
Uray, K.,
Somsák, L.,
Docsa, T.,
Bokor, É.:
Dual-Target Compounds against Type 2 Diabetes Mellitus: proof of Concept for Sodium Dependent Glucose Transporter (SGLT) and Glycogen Phosphorylase (GP) Inhibitors.
Pharmaceuticals. 14 (4), 1-27, 2021.
Kiss, M.,
Szabó, E.,
Bocska, B.,
Sinh, L. T.,
Fernandes, C. P.,
Timári, I.,
Hayes, J. M.,
Somsák, L.,
Barna, T.:
Nanomolar inhibition of human OGA by 2-acetamido-2-deoxy-d-glucono-1,5-lactone semicarbazone derivatives.
Eur. J. Med. Chem. 223, 1-14, (article identifier: 113649), 2021.