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Department of Pharmaceutical Chemistry

Department of Pharmaceutical Chemistry
Department of Pharmaceutical Chemistry
Uploaded publications:
399
Publications in DEA:
263
OA:
93
Date range:
1975-2025
2025
1.
Bege, M., Kattoub, R. G., Borbás, A.: Avacincaptad pegol, the second approved aptamer medicine: a mini review.
DRem. 1 (2), 29-45, 2025.
2.
Bege, M., Borbás, A.: New anticancer medicines approved by the EMA in 2024.
DRem. 1 (2), 46-56, 2025.
3.
Kelemen, V., Bege, M., Debreczeni, N., Bereczki, I., Bényei, A., Herczegh, P., Borbás, A.: Stereoselective Synthesis of 1,2-cis-alpha-Glycosyl Thiols and Trehalose-Type alpha,alpha'-Thiodisaccharides by Cryo Thiol-Ene Photocoupling - Thio-Click Reaction in Frozen State.
Chem.-Eur. J. [Epub ahead of print], 1-10, (article identifier: 202500104), 2025.
Journal metrics:
Q2 Catalysis (2024)
Q1 Chemistry (miscellaneous) (2024)
Q1 Organic Chemistry (2024)
4.
Bege, M., Lovas, M., Priksz, D., Bernát, B., Bereczki, I., Kattoub, R. G., Kajtár, R., Eskeif, S., Novák, L., Hodek, J., Weber, J., Herczegh, P., Lekli, I., Borbás, A.: Synthesis, H2S releasing properties, antiviral and antioxidant activities and acute cardiac effects of nucleoside 5'-dithioacetates.
Sci Rep. 15 (1), 2876-2881, 2025.
Journal metrics:
Q1 Multidisciplinary (2024)
5.
Bege, M., Leiner, K., Lovas, M., Pető, R., Bereczki, I., Hodek, J., Weber, J., Kuczmog, A., Borbás, A.: Synthesis of 3'-modified xylofuranosyl nucleosides bearing 5'-silyl or -butyryl groups and their antiviral effect against RNA viruses.
Eur. J. Pharm. Sci. 209, 1-12, (article identifier: 107107), 2025.
Journal metrics:
Q1 Pharmaceutical Science (2024)
6.
Bege, M., Kattoub, R. G., Borbás, A.: The 20th Anniversary of Pegaptanib (MacugenTM), the First Approved Aptamer Medicine: history, Recent Advances and Future Prospects of Aptamers in Therapy.
Pharmaceutics. 17 (3), 394-, 2025.
Journal metrics:
D1 Pharmaceutical Science (2024)
7.
Kútvölgyi, K., Peleskei, Z., Demeter, F., Barta, R. A., Mándi, A., Homoki, E., Oláh, A., Hajkó, J., Herczeg, M., Lisztes, E.: The First Simplified Heparan Sulphate: Alginate Hybrid Trisaccharides: Synthesis and Biological Effects on Human Dermal Fibroblasts.
Int. J. Mol. Sci. 26 (17), 1-35, (article identifier: 8305), 2025.
Journal metrics:
Q2 Catalysis (2024)
Q1 Computer Science Applications (2024)
Q1 Inorganic Chemistry (2024)
Q1 Medicine (miscellaneous) (2024)
Q2 Molecular Biology (2024)
D1 Organic Chemistry (2024)
Q1 Physical and Theoretical Chemistry (2024)
D1 Spectroscopy (2024)
2024
8.
Tósaki, Á., Szabó, Z., Király, J., Lőrincz, E. B., Vass, V., Tánczos, B., Bereczki, I., Herczegh, P., Remenyik, É., Tósaki, Á., Szabó, E.: A new cannabigerol derivative, LE-127/2, induces autophagy mediated cell death in human cutaneous melanoma cells.
Eur. J. Pharm. Sci. 203, 1-15, (article identifier: 106920), 2024.
Journal metrics:
Q1 Pharmaceutical Science
9.
Faltinek, L., Melicher, F., Kelemen, V., Mező, E., Borbás, A., Wimmerová, M.: Bispecific Thio-Linked Disaccharides as Inhibitors of Pseudomonas Aeruginosa Lectins LecA (PA-IL) and LecB (PAIIL): dual-Targeting Strategy.
Chem.-Eur. J. 30, 1-10, (article identifier: 202403546), 2024.
Journal metrics:
Q2 Catalysis
Q1 Chemistry (miscellaneous)
Q1 Organic Chemistry
10.
Herczeg, M., Demeter, F., Nagy, T., Rusznyák, Á., Hodek, J., Sipos, É., Lekli, I., Fenyvesi, F., Weber, J., Kéki, S., Borbás, A.: Block Synthesis and Step-Growth Polymerization of C-6-Sulfonatomethyl-Containing Sulfated Malto-Oligosaccharides and Their Biological Profiling.
Int. J. Mol. Sci. 25 (1), 1-29, (article identifier: 677), 2024.
Journal metrics:
Q2 Catalysis
Q1 Computer Science Applications
Q1 Inorganic Chemistry
Q1 Medicine (miscellaneous)
Q2 Molecular Biology
D1 Organic Chemistry
Q1 Physical and Theoretical Chemistry
D1 Spectroscopy
11.
Tóth, I. B., Bazeli, B., Janssens, A., Lisztes, E., Racskó, M., Kelemen, B., Herczeg, M., Nagy, T. M., Kövér, K. E., Mitra, A., Borics, A., Bíró, T., Voets, T.: Direct modulation of TRPM8 ion channels by rapamycin and analog macrolide immunosuppressants.
eLife. 13, (article identifier: 97341), 2024.
Journal metrics:
D1 Biochemistry, Genetics and Molecular Biology (miscellaneous)
D1 Immunology and Microbiology (miscellaneous)
D1 Medicine (miscellaneous)
D1 Neuroscience (miscellaneous)
12.
Tánczos, B., Vass, V., Szabó, E., Lovas, M., Kattoub, R. G., Bereczki, I., Borbás, A., Herczegh, P., Tósaki, Á.: Effects of H2S-donor ascorbic acid derivative and ischemia/reperfusion-induced injury in isolated rat hearts.
Eur. J. Pharm. Sci. 195, 1-15, (article identifier: 106721), 2024.
Journal metrics:
Q1 Pharmaceutical Science
13.
Király, J., Szabó, E., Fodor, P., Vass, A., Choudhury, M., Gesztelyi, R., Szász, C., Flaskó, T., Dobos, N., Zsebik, B., Steli, Á. J., Halmos, G., Szabó, Z.: Expression of hsa-miRNA-15b, -99b, -181a and Their Relationship to Angiogenesis in Renal Cell Carcinoma.
Biomedicines. 12 (7), 1-18, (article identifier: 1441), 2024.
Journal metrics:
Q1 Biochemistry, Genetics and Molecular Biology (miscellaneous)
Q1 Medicine (miscellaneous)
14.
Bege, M., Borbás, A.: Medicines for influencing the posttranslational modifications of histones - a tutorial review.
DRem. 1 (1), 1-13, 2024.
15.
Moreau, F., Atamanyuk, D., Blaukopf, M., Barath, M., Herczeg, M., Xavier, N. M., Monbrun, J., Airiau, E., Henryon, V., Leroy, F., Floquet, S., Bonnard, D., Szabla, R., Brown, C., Junop, M. S., Kosma, P., Gerusz, V.: Potentiating Activity of GmhA Inhibitors on Gram-Negative Bacteria.
J. Med. Chem. 67 (8), 6610-6623, 2024.
Journal metrics:
D1 Drug Discovery
Q1 Molecular Medicine
16.
Hőgye, F., Farkas, L. B., Balogh, Á. K., Szilágyi, L., Samar, A., Bajza, I., Borbás, A., Fehér, K., Illyés, T. Z., Timári, I.: Saturation Transfer Difference NMR and Molecular DockingInteraction Study of Aralkyl-Thiodigalactosides as Potential Inhibitors of the Human-Galectin-3 Protein.
Int. J. Mol. Sci. 25 (3), 1-18, (article identifier: 1742), 2024.
Journal metrics:
Q2 Catalysis
Q1 Computer Science Applications
Q1 Inorganic Chemistry
Q1 Medicine (miscellaneous)
Q2 Molecular Biology
D1 Organic Chemistry
Q1 Physical and Theoretical Chemistry
D1 Spectroscopy
17.
Demeter, F., Peleskei, Z., Kútvölgyi, K., Rusznyák, Á., Fenyvesi, F., Kajtár, R., Sipos, É., Lekli, I., Molnár, P., Szöllősi, A. G., Lisztes, E., Tóth, I. B., Borbás, A., Herczeg, M.: Synthesis and Biological Profiling of Seven Heparin and Heparan Sulphate Analogue Trisaccharides.
Biomolecules. 14 (9), 1-24, (article identifier: 1052), 2024.
Journal metrics:
Q1 Biochemistry
Q2 Molecular Biology
18.
Bege, M., Borbás, A.: The Design, Synthesis and Mechanism of Action of Paxlovid, a Protease Inhibitor Drug Combination for the Treatment of COVID-19.
Pharmaceutics. 16 (2), 1-17, (article identifier: 217), 2024.
Journal metrics:
D1 Pharmaceutical Science
19.
Óvári, I., Viczján, G., Bege, M., Borbás, A., Herczegh, P., Zsuga, J., Papp, Z., Szilvássy, Z., Juhász, B., Gesztelyi, R., Erdei, T. D.: The ex vivo effects of hypoxanthine-tricyclano, a synthetic adenosine analogue, on rat left and right atria.
Gen. Physiol. Biophys. 43 (6), 577-584, 2024.
Journal metrics:
Q3 Biophysics
Q3 Medicine (miscellaneous)
Q4 Physiology
2023
20.
Godoy, A. S., Nakamura, A. M., Douangamath, A., Song, Y., Noske, G. D., Gawriljuk, V. O., Fernandes, R. S., Pereira, H. D. M., Oliveira, K. I. Z., Fearon, D., Dias, A., Krojer, T., Fairhead, M., Powell, A., Dunnet, L., Brandao-Neto, J., Skyner, R., Chalk, R., Bajusz, D., Bege, M., Borbás, A., Keserű, G. M., Delft, F. v., Oliva, G.: Allosteric regulation and crystallographic fragment screening of SARS-CoV-2 NSP15 endoribonuclease.
Nucleic Acids Res. 51 (10), 5255-5270, 2023.
Journal metrics:
D1 Genetics
21.
Lőrincz, E. B., Herczeg, M., Houser, J., Rievajová, M., Kuki, Á., Malinovská, L., Naesens, L., Wimmerová, M., Borbás, A., Herczegh, P., Bereczki, I.: Amphiphilic Sialic Acid Derivatives as Potential Dual-Specific Inhibitors of Influenza Hemagglutinin and Neuraminidase.
Int. J. Mol. Sci. 24, 1-23, (article identifier: 17268), 2023.
Journal metrics:
Q2 Catalysis
Q1 Computer Science Applications
D1 Inorganic Chemistry
Q1 Medicine (miscellaneous)
Q2 Molecular Biology
D1 Organic Chemistry
Q1 Physical and Theoretical Chemistry
D1 Spectroscopy
22.
Farkas, G., Császár, Z., Tóth-Farsang, E., Bényei, A., Bakos, J.: Application of alkane-diyl based chiral phosphine-aminophosphine (P-NP) and thioether-aminophosphine (S-NP) ligands in Rh-catalyzed asymmetric hydrogenation.
J. Organomet. Chem. 994, 1-8, (article identifier: 122723), 2023.
Journal metrics:
Q3 Biochemistry
Q3 Inorganic Chemistry
Q3 Materials Chemistry
Q3 Organic Chemistry
Q3 Physical and Theoretical Chemistry
23.
Fésüs, A., Ábrahám, A., Sipos, É., Szőke, K., Bak, I., Kiss-Szikszai, A., Lekli, I.: Evaluation of the antioxidant effect of kd15 and kd36 newly synthetized molecules.
In: FAMÉ 2023 Mátraháza 7-9 June 2023 : Programme Oral and Poster Abstract / org. Hungarian Society For Experimental And Clinical Pharmacology, Hungarian Physiological Society, Hungarian Society For Microcirculation And Vascular Biology, HUPHAR, [S.l.], 223, 2023.
24.
Demeter, F., Török, P., Kiss, A., Kovásznai-Oláh, R., Máthéné Szigeti, Z., Baksa, V., Kovács, F., Balla, N., Fenyvesi, F., Váradi, J., Borbás, A., Herczeg, M.: First Synthesis of DBU-Conjugated Cationic Carbohydrate Derivatives and Investigation of Their Antibacterial and Antifungal Activity.
Int. J. Mol. Sci. 24 (4), 1-20, (article identifier: 3550), 2023.
Journal metrics:
Q2 Catalysis
Q1 Computer Science Applications
D1 Inorganic Chemistry
Q1 Medicine (miscellaneous)
Q2 Molecular Biology
D1 Organic Chemistry
Q1 Physical and Theoretical Chemistry
D1 Spectroscopy
25.
Chniti, S., Kollár, L., Bényei, A., Dörnyei, Á., Takács, A.: Highly Chemoselective One-Step Synthesis of Novel N- Substituted-Pyrrolo[3,4-b]quinoline-1,3-diones via Palladium-Catalyzed Aminocarbonylation/Carbonylative Cyclisation Sequence.
Eur. J. Org. Chem. 26 (10), 1-8, (article identifier: 202201374), 2023.
Journal metrics:
Q2 Organic Chemistry
Q2 Physical and Theoretical Chemistry
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